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Search Results for " lysine-specific demethylase 1 inhibitor "

20

Compounds

Cat No. Product Name Synonyms Targets
T6835 Fenoldopam mesylate Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526 Dopamine Receptor
Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties. It lowers blood pressure through arteriolar vasodilation.
T7942 Tranylcypromine hemisulfate Tranylcypromine Sulfate,Tranylcypromine (hemisulfate) Histone Demethylase , MAO , Monoamine Oxidase
Tranylcypromine hemisulfate (Tranylcypromine Sulfate) is an inhibitor of monoamine oxidase (MAO) and lysine-specific demethylase 1 (LSD1) with a rapid onset of activity.
T4418 GSK2879552 2HCl (1401966-69-5(free base)) Histone Demethylase
GSK2879552 is an orally available, irreversible inhibitor of lysine specific demethylase 1 (LSD1), with potential antineoplastic activity.
T21652 RN-1 dihydrochloride Histone Demethylase , MAO
RN-1 dihydrochloride is an effective and selective irreversible inhibitor of lysine-specific demethylase 1 (LSD1, IC50 = 70 nM).
T83966 LSD1-IN-30 Histone Demethylase
LSD1-IN-30 is a lysine-specific demethylase 1 (LSD1) inhibitor with anticancer activity for the study of small cell lung cancer and acute myeloid leukemia.
T11882 Pulrodemstat benzenesulfonate LSD1-IN-7 benzenesulfonate,CC-90011 benzenesulfonate Histone Demethylase
Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
T4477 Domatinostat tosylate 4SC-202 tosylate,4SC-202 Apoptosis , HDAC
Domatinostat tosylate (4SC-202) is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
T6362 Domatinostat 4SC202,4SC 202,4SC-202 (free base),4SC-202 Apoptosis , HDAC
Domatinostat (4SC202) is a selective class I HDAC inhibitor with IC50 of 1.20 μM, 1.12 μM, and 0.57 μM for HDAC1, HDAC2, and HDAC3, respectively. Also displays inhibitory activity against Lysine specific demethylase 1 (L...
T39252L 5-[(1S,2S)-2-[(Cyclopropylmethyl)amino]cyclopropyl]-N-(tetrahydro-2H-pyran-4-yl)thiophene-3-carboxamide hydrochloride Others
5-[(1S,2S)-2-[(Cyclopropylmethyl)amino]cyclopropyl]-N-(tetrahydro-2H-pyran-4-yl)thiophene-3-carboxamide hydrochloride is a cyclopropanoid enzyme compound that acts as a lysine-specific demethylase-1 inhibitor for schizop...
T13057 T-448 Histone Demethylase
T-448 is a specific, orally active and irreversible lysine-specific demethylase 1 (LSD1, an H3K4 demethylase) inhibitor(IC50 of 22 nM).
T13056 T-448 free base Histone Demethylase
T-448 free base is a specific, orally active and irreversible lysine-specific demethylase 1 (LSD1, an H3K4 demethylase) inhibitor(IC50 of 22 nM).
T11883 Pulrodemstat Methylbenzenesulfonate LSD1-IN-7 Methylbenzenesulfonate Others
LSD1-IN-7 Methylbenzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
T13052 S2101 S 2101 Histone Demethylase
S 2101 is an inhibitor of lysine-specific demethylase 1 (LSD1)(IC50 of 0.99 μM, Ki of 0.61 μM and Kinact/Ki of 4560 M/s).
T11880 LSD1-IN-5 Histone Demethylase
LSD1-IN-5 increases dimethylated Lys4 of histone H3, shows no effect on expression of LSD1. LSD1-IN-5 is a potent and reversible inhibitor of lysine-specific demethylase 1 (LSD1), with an IC50 of 121 nM.
T39226 INCB059872 INCB059872
INCB059872 is a highly potent, orally active, selective, and irreversible inhibitor of Lysine-Specific Demethylase 1 (LSD1). Its chemical properties make it suitable for use in researching myeloid leukemia.
T11881 LSD1-IN-6 Histone Demethylase
LSD1-IN-6 increases dimethylated Lys4 of histone H3, shows no effect on expression of LSD1. LSD1-IN-6 is a potent and reversible inhibitor of lysine-specific demethylase 1 (LSD1), with an IC50 of 123 nM.
T40420 Namoline
Namoline is a γ-pyrone compound that functions as a selective and reversible inhibitor of Lysine-specific demethylase 1 (LSD1) with an IC50 of 51 μM in an HRP-coupled enzymatic assay. By impairing LSD1 demethylase activi...
T61565 KDM5B-IN-3
KDM5B-IN-3 (Compound 5) is an inhibitor of histone lysine-specific demethylase 5B (KDM5B) or JARID1B. It effectively inhibits the activity of KDM5B with an IC50 value of 9.32 μM. Consequently, KDM5B-IN-3 serves as a valu...
T36625 LSD1/HDAC6-IN-1 LSD1/HDAC6-IN-1
LSD1/HDAC6-IN-1 is an orally active compound that functions as a dual inhibitor, targeting lysine specific demethylase 1 (LSD1) and histone deacetylase 6 (HDAC6). This compound demonstrates promising anti-tumor activity ...
T11503 GSK 690 Hydrochloride Histone Demethylase
GSK 690 (Hydrochloride) is a reversible lysine specific demethylase 1 (LSD1) inhibitor with a Kd value of 9 nM and IC 50 of 37 nM.

Compounds

Fenoldopam mesylate
T6835
Synonym: Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526
Target: Dopamine Receptor
Tranylcypromine hemisulfate
T7942
Synonym: Tranylcypromine Sulfate,Tranylcypromine (hemisulfate)
Target: Histone Demethylase, MAO, Monoamine Oxidase
GSK2879552 2HCl (1401966-69-5(free base))
T4418
Synonym:
Target: Histone Demethylase
RN-1 dihydrochloride
T21652
Synonym:
Target: Histone Demethylase, MAO
LSD1-IN-30
T83966
Synonym:
Target: Histone Demethylase
Pulrodemstat benzenesulfonate
T11882
Synonym: LSD1-IN-7 benzenesulfonate,CC-90011 benzenesulfonate
Target: Histone Demethylase
Domatinostat tosylate
T4477
Synonym: 4SC-202 tosylate,4SC-202
Target: Apoptosis, HDAC
Domatinostat
T6362
Synonym: 4SC202,4SC 202,4SC-202 (free base),4SC-202
Target: Apoptosis, HDAC
5-[(1S,2S)-2-[(Cyclopropylmethyl)amino]cyclopropyl]-N-(tetrahydro-2H-pyran-4-yl)thiophene-3-carboxamide hydrochloride
T39252L
Synonym:
Target: Others
T-448
T13057
Synonym:
Target: Histone Demethylase
T-448 free base
T13056
Synonym:
Target: Histone Demethylase
Pulrodemstat Methylbenzenesulfonate
T11883
Synonym: LSD1-IN-7 Methylbenzenesulfonate
Target: Others
S2101
T13052
Synonym: S 2101
Target: Histone Demethylase
LSD1-IN-5
T11880
Synonym:
Target: Histone Demethylase
INCB059872
T39226
Synonym: INCB059872
Target:
LSD1-IN-6
T11881
Synonym:
Target: Histone Demethylase
Namoline
T40420
Synonym:
Target:
KDM5B-IN-3
T61565
Synonym:
Target:
LSD1/HDAC6-IN-1
T36625
Synonym: LSD1/HDAC6-IN-1
Target:
GSK 690 Hydrochloride
T11503
Synonym:
Target: Histone Demethylase
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TargetMol